Custom Peptides
Cayman Chemical 2-Ethylamino-1-phenylbutane (hydrochloride), Purity: ≥98%, CAS: 29805-52-5, 10 mg
An analog of N-ethylamphetamine that is characterized by an ethyl group replacing methyl at the α position
Cayman Chemical Cintirorgon, Purity: ≥98%, CAS: 2055536-64-4, 10 mg
A RORɣ agonist (EC50s = <0.5 µM in a reporter assay and TR-FRET assay)
Cayman Chemical AurothIoglucosehydrate 10mg
A TrxR inhibitor (IC50 = 0.065 µM for the human placental enzyme); selective for TrxR over glutathione reductase and GPX (IC50s = >100 and 80 µM, respectively); inhibits IL-1β-induced production of IL-6 and IL-8 in isolated human rheumatoid synovial fibroblasts at 100 µM; reduces HIV-1 replication induced by TNF-α in OM10.1 cells latently infected with HIV-1 at 10 and 25 µM; improves survival in a mouse model of ARDS induced by LPS and hyperoxia at 25 mg/kg; induces obesity and increases food intake and blood glucose levels in genetically diabetic KK mice
Cayman Chemical Ursocholic Acid, Purity: ≥95%, CAS: 2955-27-3, 10 mg
A bile acid; dietary administration decreases gallbladder cholesterol, phospholipid, and bile acid levels and the occurrence of gallstones in male mice fed a lithogenic diet at 0.25%
Cayman Chemical 16-Oxokahweol, Purity: ≥98%, CAS: 108664-99-9, 10 mg
A synthetic diterpene; increases cytosolic GST activity and acid-soluble sulfhydryl levels in mouse liver and small bowel mucosa at 10 µmol once per day for three days
Cayman Chemical 5fluoro MPPICA phnylpropI 10mg
An analytical reference standard that is structurally similar to known synthetic cannabinoids; a potential metabolite of 5-fluoro MPP-PICA based on the published metabolism of 5-fluoro AMB-PICA; intended for research and forensic applications
Cayman Chemical Chamazulene, Purity: ≥98%, CAS: 529-05-5, 10 mg
A terpene with anti-inflammatory and antioxidant activities; reduces increases in MMP-3, MMP-9, COX-2, iNOS, and p65 NF-κB levels in IL-1β-stimulated primary rat chondrocytes at 10 µg/ml; reduces IL-1β-induced production of MDA and increases levels of SOD, catalase, and GPX in primary rat chondrocytes at 10 and 20 µg/ml; reduces hind paw volume, serum levels of MDA, TNF-α, and IL-6, and cartilage erosion in a rat model of CFA-induced osteoarthritis at 25 and 50 mg/kg
Cayman Chemical Boc-Glu-OBzl, Purity: ≥98%, CAS: 30924-93-7, 5 g
An amino acid building block; has been used in the synthesis of peptide-based inhibitors of human caspases and HRV 3C protease that have enzyme inhibitory activity in vitro
Cayman Chemical Wilforgine, Purity: ≥98%, CAS: 37239-47-7, 10 mg
A sesquiterpene alkaloid with paralytic activity; induces paralysis in third instar M. separata larvae (NC50 = 0.0086 µmol/larvae)
Cayman Chemical ParasIn IcatfIshtrIfluor 10mg
An antimicrobial peptide; active against various Gram-positive and Gram-negative bacteria, as well as fungi (MICs = 1-2, 1-4, and 1-2 UG/ml, respectively)
Cayman Chemical 5,6-dihydro-5-Fluorouracil, Purity: ≥95%, CAS: 696-06-0, 10 mg
An active metabolite of 5-fluorouracil; is cytotoxic to HaCaT cells (IC50 = 13.5 µM); reduces tumor growth in combination with 5-fluorouracil and eniluracil in a rat model of colon carcinoma at 90 mg/kg per week
Cayman Chemical 3-Methylbuphedrone (hydrochloride), Purity: ≥98%, CAS: 1797911-07-9, 10 mg
A methylated analog of buphedrone; intended for forensic and research applications
Cayman Chemical 4'-O-methyl Quercetin, Purity: ≥95%, CAS: 603-61-2, 10 mg
A flavonoid from C. ordata with anticancer and antiplasmodial activity; inhibits the viability of HL-60, U937, MOLT-3, Raji, K562, MCF-7, SK-MEL-1, and A549 human tumor cell lines with IC50 values ranging from 5.5-24.1 μM; induces G2-M arrest and inhibits tubulin polymerization in vitro; inhibits breast cancer resistance protein (BCRP/ABCG2; IC50 = 0.040 μM in a vesicular transport assay); reduces in vitro proliferation of chloroquine-resistant P. falciparum (IC50 = 4.8 μM)